Ofloxacin shahararren magani ne saboda yana da alamomi masu yawa don amfani, kuma an tabbatar da ingancin warkewar magani ba kawai ta hanyar karatun asibiti ba, har ma da kwarewar marasa lafiya.
Sunan kasa da kasa
Ana amfani da samfurin magunguna a duk duniya. An rubuta sunan ƙasa da ƙasa cikin Latin kamar Ofloxacin.
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Ofloxacin shahararren magani ne.
ATX
Dangane da ilimin halittar jiki, warkewa da rarrabuwa masu guba, ƙwayar tana nufin magungunan antimicrobial na aikin tsari. Wannan rukunin ya ƙunshi wakilai masu hana ƙwayoyin cuta aiki na tsarin aiki. Wadannan sun hada da quinolones da fluoroquinolones, wadanda suka hada magunguna. An sanya masa lambar ATX: J01MA01.
Saki siffofin da abun da ke ciki
Wannan samfurin yana da nau'ikan iri, wanda kowannensu ke nufi don amfanin ciki ko na gida. Babban sinadari mai aiki a cikin dukkan nau'ikan magungunan shine wani abu mai haɓaka wanda ke ba da sunan kasuwanci.
Cutar rigakafi ce mai yawan gaske. Yana da tasiri a kan manyan adadin cututtukan ƙwayoyin cuta. Componentsarin abubuwan da aka gyara ba su da tasirin warkewa kuma suna yin ayyuka na taimako.
Kwayoyi
Allunan suna da siffar biconvex zagaye. Fim mai ruɓi yana narkewa cikin sauƙi. Launin maganin ya kusan fari. Sashi na 1 na kwayoyin zai iya zama 200 ko 400 MG na kayan aiki. Ana ɗaukar allunan a baka. An tattara magungunan a cikin blisters da kwali na fakiti.
Magani
Ana samun wakilin antibacterial a cikin hanyar maganin jiko. An sanya magani mai launin rawaya a cikin gilashin gilashin giram 100 ml. Baya ga abu mai aiki, abun da ke cikin maganin ya hada da sinadarin sodium chloride da ruwa mai tsafta don yin allura. 100 ml na mafita ya ƙunshi 2 g na kayan aiki mai aiki.
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Maganin shafawa
Maganin shafawa an yi shi ne domin magance cututtukan ido. An samar da shi a cikin bututu na aluminium na 3 ko 5 g. Haɗin maganin ya haɗa da ƙwayar roba, har da tsofaffin abubuwa: petrolatum, nipagin, gamezole. Maganin shafawa yana da farin ko launin shuɗi mai launin shuɗi da tsarin tsari.
Aikin magunguna
Ma'aikacin kantin magani yana da ikon dakatar da kira na wani enzyme wanda ya dace don inganta DNA na nau'ikan masu kamuwa da cuta. Lalacewa mahimman abubuwan jikin kwayar halitta suna haifar da mutuwarsa. Saboda haka, miyagun ƙwayoyi yana da maganin antimicrobial da sakamako na kwayan cuta.
Kwayar rigakafi tana da inganci a kan ƙananan ƙwayoyin cuta waɗanda ke samar da beta-lactamases. Magungunan zai iya magance cutar mycobacteria da ke saurin girma. Magungunan, mallakar ƙarni na 2 na fluoroquinolones, yana da rawar da za ta iya ɗauka game da microflora gram-positive da gram-korau.
Kwayoyin cutar anaerobic sune yawancin ƙwayoyin cuta. Treponema pallidum ba shi da kula da maganin.
Pharmacokinetics
Abubuwan da ke cikin manyan abubuwan suna haɗuwa cikin jini cikin hanzari daga narkewa kuma ana kusan kasancewa cikin jiki. Abubuwan da ke aiki suna shiga cikin sel na gabobin ciki, gami da waɗanda ke da alaƙa da tsarin numfashi, urinary da tsarin haihuwa.
Kwayoyin rigakafi suna tarawa cikin dukkan ruwayen jiki, guringuntsi da gidajen abinci.
Ana lura da mafi girman yawan hankali bayan kimanin minti 60. Kusan kashi 5% na miyagun ƙwayoyi suna cikin metabolized a cikin hanta. Cire rabin rayuwar shine 6-7 hours. Kusan 80-90% na abu mai aiki an cire shi daga jiki ta hanyar kodan, karamin sashi - tare da bile.
Menene taimaka?
Wideaƙƙarfan aiki da yawa na ƙaddara aikin aikace-aikacen antimicrobial wanda zai iya yaƙi da cututtukan ƙwayar cuta na ƙananan wurare daban-daban. An wajabta magungunan ga cututtuka irin su:
- kumburi da tsakiyar kunne, sinusitis, sinusitis, gaban sinusitis;
- cutar kuturta da ke rufe hanji da kumburin ciki (cystitis, urethritis, pyelonephritis);
- cututtukan ƙwayar cuta na ƙwayar ciki;
- cututtukan kumburi daga cikin mahaifa da tsarin na huhu (pharyngitis, laryngitis, pneumonia);
- pathologies na fata da lalacewar kyallen takarda mai kaushi, kasusuwa da gidajen abinci da ke hade da haɓakar microflora na pathogenic;
- cututtukan cututtukan ƙwayar cuta da cututtukan ƙwayar cuta na jiki (colpitis, endometritis, prostatitis, cervicitis, salpingitis);
- cututtukan cututtukan mahaifa na cornea, conjunctivitis, blepharitis, dacryocystitis, sha'ir, cututtukan ido da chlamydia ta haifar.
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Ana amfani da maganin rigakafi sau da yawa kafin tiyata don hana rikicewa bayan tiyata.
Contraindications
Ba za a iya amfani da maganin tare da ƙara yawan ji da ƙwaƙwalwa da daidaituwa na mutum zuwa abubuwan da aka gyara ba. An haramta duk nau'ikan fitarwa yayin daukar ciki, lokacin shayarwa da kuma a cikin yara 'yan ƙasa da shekaru 18. A cikin cututtukan zuciya da ƙwaƙwalwar ƙwayar cuta, mummunan cututtukan hanta da hanta, kodan da zuciya, ƙwayar rigakafi tana karɓa. Lalacewar latose da lalacewar jiji yayin shan magunguna daga ƙungiyar fluoroquinolone suna buƙatar zaɓi wani wakili don kula da kamuwa da cuta.
Yadda za a ɗauka?
Shawarar shan magani, nau'ikan sashi, sashi da tsawon lokacin amfani da miyagun ƙwayoyi an ƙaddara ta likita dangane da tsananin cutar, shekarun mai haƙuri da alaƙa da cutar.
Kafin ko bayan abinci?
Allunan ana ɗauka kafin ko lokacin abinci, suna haɗiye su gaba ɗaya. Adadin yau da kullun ga manya shine 200-800 mg kuma an kasu kashi biyu. Tsawon lokacin aikin shine 5-10 kwana. Dole ne a dauki maganin a cikin kwanaki 3 bayan ɓacewar manyan alamun cutar.
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Ana sarrafa maganin allurar sau ɗaya don rabin sa'a. Sashi shine 200 MG. Tare da haɓakawa a cikin hoto na asibiti, sannan sai a tura mai haƙuri zuwa maganin ƙwayoyin cuta na baka. Idan ya cancanta, bayar da allurar ciki na 100-200 MG sau 2 a rana. Ga mutanen da ke da ƙarancin rigakafin cutar, ana iya ninka sashi zuwa 500 MG kowace rana.
Ana maganin cututtukan Chlamydial na idanu tare da maganin shafawa: 1 cm (kimanin 2 MG) na miyagun ƙwayoyi an sanya shi cikin jakar haɗuwa daga sau 3 zuwa 5 a rana.
Shin yana yiwuwa a sha maganin don ciwon sukari?
Marasa lafiya waɗanda ke fama da ciwon sukari an basu damar ɗaukar magani a ƙarƙashin yanayin kula da kullun matakan glucose jini. Magungunan rigakafi tare da insulin na iya haifar da cutar hypoglycemia mai ƙarfi. Kafin fara amfani da shi, ya zama dole a nemi likita kuma a ba da rahoto game da magunguna da mutum ya ɗauka a kan ci gaba.
Side effects
Fluoroquinolones na iya haifar da mummunan sakamako masu illa, alamun farko waɗanda ya kamata su daina shan kwayoyin kuma ku shawarci likitan ku don sake nazarin tsarin kula da cutar don kamuwa da cuta.
Gastrointestinal fili
Magungunan a wasu yanayi na haifar da tashin zuciya, amai, zawo. Ci gaban cholestatic jaundice, pseudomembranous enterocolitis, da haɓaka ayyukan hepatic transaminases ba su yanke hukunci ba. Sau da yawa marasa lafiya suna koka da zafi da rashin jin daɗi a cikin ƙoshin ciki.
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Hematopoietic gabobin
Magani ya keta alamun asibiti na jini kuma yana iya zama sanadiyyar anemia, agranulocytosis, leukopenia, thrombocytopenia.
Tsarin juyayi na tsakiya
Daga gefen tsarin juyayi na tsakiya, haɓakar rashin ƙarfi da narkewa, daidaitaccen daidaituwa na motsi, an lura da asarar ji. A wasu halaye, mutum ya sami ƙara damuwa da tsoro. Rashin damuwa, rashin bacci ko raye-raye a cikin mafarki, ba a cire musu fahimta launi.
Daga tsarin urinary
Wani wakili na antibacterial na iya kara urea kuma yana haifar da matsanancin ƙwaƙwalwar ƙwayar cuta. Ya kamata a kula da allunan tare da taka tsantsan, tunda lalacewar koda na iya faruwa.
Daga tsarin numfashi
Sakamakon sakamako na gefe daga tsarin numfashi yana bayyana a cikin hanyar bushe tari, bronchospasm da tsananin numfashi.
Daga tsarin musculoskeletal
Tasiri mara kyau akan tsarin musculoskeletal da tsarin musculoskeletal shine bayyanar alamun bayyanar myalgia, arthralgia. Ba a cire Tendon rupture ba, musamman ma a cikin tsofaffi marasa lafiya.
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Daga tsarin zuciya
Magungunan ƙwayar ƙwayar cuta na iya lalata aikin zuciya. An yi rikodin lokuta na tachycardia, bradycardia, vasculitis da rushewa.
Cutar Al'aura
Abubuwan da suka fi yawan tasirin sakamako sune halayen rashin lafiyan, kamar itching, redness na saman layuka na epidermis, fatar fata, urticaria, anaphylactic shock, Quincke's edema.
Umarni na musamman
Ba a yi amfani da kayan aikin don magance cututtukan ƙwayar cuta mai narkewa da ciwon huhu da tsokanar ƙwayar cuta ta pneumococci ba. Ana buƙatar daidaita sikelin don cututtukan cututtukan zuciya masu ƙarfi na zuciya, hanta da kodan.
Idan allunan tsokanan pseudomembranous enterocolitis, metronidazole ya kamata a wajabta su ga mai haƙuri.
Kada a sha kwayoyin rigakafi fiye da kwanaki 60. Yayin jiyya, ana bada shawara don guje wa radiation na ultraviolet.
Amfani da barasa
Kada a yi amfani da magani a cikin haɗuwa tare da barasa. Barasa yana inganta tasirin mai guba na abubuwan da ke tattare da ƙwayar cuta kuma yana tsokani ci gaban mummunan sakamako masu illa.
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Tasiri kan ikon sarrafa abubuwan inji
Magungunan yana rage jinkirin halayen psychomotor na jiki, mummunar rinjayar ikon fitar da motoci da ƙananan hanyoyin. Sabili da haka, mutanen da ke aiki da masana'antu masu fasaha na haɗari masu haɗari da direbobi a yayin da ya kamata suyi hankali sosai.
Yi amfani da lokacin daukar ciki da lactation
Abubuwa masu aiki suna shiga katangar mahaifa kuma ke cutar da tayin na ciki. Abubuwan da ke tattare da rigakafin sun kasance a cikin madara, wadanda zasu cutar da lafiyar jariri. A lokacin daukar ciki da lactation, maganin yana contraindicated. Idan uwa mai shayarwa tana buƙatar yin aikin tiyata, an koma da yaron zuwa abinci mai wucin gadi.
Yi amfani da tsufa
A cikin tsufa, ana wajabta maganin don dalilai na kiwon lafiya. Ana gudanar da maganin a ƙarƙashin kulawar likita. Kwayoyin kwayoyi suna tsoratar da jijiyoyin jiki a cikin tsofaffi marasa lafiya.
Yawan damuwa
Wucewa yawan maganin da aka yarda da shi yana haifar da ci gaban tashin zuciya da amai, rashin daidaituwa da motsi, rikicewa, ciwon kai da bushewar baki. Babu takamaiman maganin rigakafi, don haka ana bai wa marasa lafiya da alamun cutar yawan ƙwayar cutar ƙwayar cuta ciki da jijiyoyin jini.
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Wucewa ƙimar maganin da aka yarda da shi yana haifar da cin zarafin daidaituwa da motsi da ciwon kai.
Yin hulɗa tare da wasu kwayoyi
A cikin cututtukan cututtuka masu raɗaɗi da kumburi, ana amfani dashi a hade tare da Ornidazole don haɓaka sakamako na antibacterial. Ba'a ba da shawarar a haɗu tare da magungunan anticoagulants na yau da kullun da magungunan cututtukan jini ba, tunda ana iya inganta aikin su. Methotrexate yana shafar narkewar tubular fluoroquinolones, yana ƙara yawan abubuwan da suke da guba.
Amfani da ciki tare da glucocorticosteroids yana kara haɗarin kamuwa da ciwon jijiyoyi, musamman a cikin tsofaffi marasa lafiya.
Antacids da kwayoyi dauke da baƙin ƙarfe, potassium, magnesium, aluminium da lithium, hulɗa tare da abubuwan da ke aiki, suna samar da mahaɗar insoluble Ya kamata a yi hutu tsakanin liyafar ire-iren waɗannan magunguna.
Amfani da haɗin gwiwa tare da magungunan anti-mai kumburi ba da shawarar ba don guje wa tasirin neurotoxic.
Analogs
Akwai magunguna da yawa na suna iri ɗaya, sunayen waɗanda suke bambanta kawai ta hanyar kari wanda ke nuna mai ƙira (Teva, Vero, FPO, Promed, ICN, Darnitsa). Waɗannan samfuran magunguna suna da kaddarorin warkewa iri ɗaya da kayan aiki 1 masu aiki.
Bugu da ƙari, kwayoyi daga jerin fluoroquinolone sune analogues na ƙwayoyin rigakafi. Yana yiwuwa a maye gurbin miyagun ƙwayoyi tare da Norfloxacin, Levofloxacin, Ciprolet. A wasu halayen, an tsara maganin rigakafi a cikin allunan ko ampoules daga wasu ƙungiyoyi: Augmentin, Amoxicillin, Rulid. Amma ya fi kyau kada ku ba da magani ga kanku, kuma a farkon alamun cutar ciwon kai, nemi likita.
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Magunguna kan bar sharuɗan
An ba da maganin kashe kwayoyin cuta tare da takardar sayan magani.
Nawa ne Ofloxacin?
Farashin magani ya dogara da nau'in sakin da wanda ya ƙera. Samfuran cikin gida suna da arha fiye da waɗancan ƙasashen waje. A cikin Ukraine, za'a iya siyan allunan don hryvnias 11.55; a cikin Rasha, farashin magani kusan 30-40 rubles.
Yanayin ajiya na miyagun ƙwayoyi Ofloxacin
Ya kamata a adana maganin a cikin busassun wuri da duhu mara izini ga yara a yawan zafin jiki.
Ranar karewa
Dole ne a yi amfani da maganin a cikin shekaru 2 daga ranar da aka nuna akan kunshin.
Binciken Ofloxacin
Vladislav, dan shekara 51, Rostov-on-Don.
Anyi maganin Ofloxacin kafin ayi tiyata ga koda koda. Abubuwan da aka fahimta sun kasance marasa kyau: ciwon kai na kullun, mara amfani mara nauyi, tashin zuciya. Amma rikice-rikice bayan tiyata bai tashi ba. Ban sani ba, allura ta taimaka, ko ba tare da su ba komai ya tafi lafiya.
Fatima, shekara 33, Nalchik.
Tare da wuce gona da iri na cystitis, Na ɗauki Allunan don 5 kwanaki. Kwayoyin cutar sun riga sun wuce aikace-aikacen 2-3. Babu wani sakamako masu illa. Magungunan suna da arha, amma yana aiki da sauri da kuma tasiri.
Stanislav, dan shekara 25, Khabarovsk.
Idanu na da ruwa da kuma farji. Ya juya cewa ya "kama" kamuwa da cuta. Anyi zubarda ido tare da Ofloxacin. Cutarwar rana tayi kwana 3.